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Cholestyramine

Cholestyramine 378GM of 4GM/DOSE

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What is Cholestyramine?

Cholestyramine is a bile acid sequestrant primarily used to lower cholesterol levels in the blood, particularly low-density lipoprotein (LDL) cholesterol. It works by binding to bile acids in the intestine, which are then excreted from the body, prompting the liver to convert more cholesterol into bile acids, thereby reducing circulating cholesterol. Additionally, cholestyramine can be used to relieve itching associated with certain liver diseases and to treat diarrhea resulting from bile acid malabsorption.

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What is Cholestyramine ?

Cholestyramine is a bile acid sequestrant primarily used to lower cholesterol levels in the blood, particularly low-density lipoprotein (LDL) cholesterol. It works by binding to bile acids in the intestine, which are then excreted from the body, prompting the liver to convert more cholesterol into bile acids, thereby reducing circulating cholesterol. Additionally, cholestyramine can be used to relieve itching associated with certain liver diseases and to treat diarrhea resulting from bile acid malabsorption.
  • Constipation
  • Stomach pain
  • Bloating
  • Gas
  • Nausea
  • Vomiting
  • Loss of appetite
  • May interfere with absorption of other medications
  • Not recommended for individuals with complete biliary obstruction
  • Caution in patients with pre-existing constipation
  • Potential for vitamin deficiency with long-term use
  • Should not be used in people with hypersensitivity to the drug
What is cholestyramine used for? ▼
Cholestyramine is FDA-approved to lower high LDL ("bad") cholesterol in primary high cholesterol, used together with a healthy diet, and to relieve itching caused by partial blockage of the bile ducts. It is a bile acid sequestrant that binds bile acids in the gut. Your doctor can tell you why it was prescribed for you.
How long does it take for cholestyramine to work? ▼
For cholesterol, cholestyramine works gradually, and it usually takes several weeks of regular use before your LDL cholesterol drops meaningfully, with your doctor rechecking levels to gauge the effect. When it is used to relieve itching from partial biliary obstruction, some people notice improvement sooner. Keep taking it as directed even if you do not feel a difference right away.
What are the most common side effects of cholestyramine? ▼
The most common side effect is constipation, which can sometimes be severe. Other common effects include bloating, gas, abdominal pain, and nausea. With long-term or high-dose use, it can lower absorption of fat-soluble vitamins (A, D, E, K) and folic acid. Contact your healthcare provider if side effects are bothersome or persistent.
Can cholestyramine be used for diarrhea and bile acid malabsorption? ▼
Cholestyramine's FDA-approved uses are lowering LDL cholesterol and relieving itching from partial biliary obstruction. Some clinicians also use it off-label for diarrhea related to bile acid malabsorption, but that is a decision only your own prescriber can make based on your situation. Do not start it for this purpose on your own; talk with your doctor.
What medications should not be taken with cholestyramine? ▼
Cholestyramine can bind many oral drugs and reduce their absorption, including thyroid hormone, warfarin, digoxin, thiazide diuretics, and some antibiotics. To avoid this, most guidance is to take your other medications at least 1 hour before or 4 to 6 hours after cholestyramine. Give your pharmacist a full list of your medicines so they can help you time doses safely.
What is Cholestyramine used for? ▼
Cholestyramine is a bile acid sequestrant primarily used to lower cholesterol levels in the blood, particularly low-density lipoprotein (LDL) cholesterol. It works by binding to bile acids in the intestine, which are then excreted from the body, prompting the liver to convert more cholesterol into bile acids, thereby reducing circulating cholesterol. Additionally, cholestyramine can be used to relieve itching associated with certain liver diseases and to treat diarrhea resulting from bile acid malabsorption.
How much does Cholestyramine cost without insurance? ▼
The price of Cholestyramine without insurance varies by pharmacy, dosage, and quantity. Rx.com compares cash prices at more than 60,000 US pharmacies so you can find the lowest price near you. Many people save up to 43% off retail prices with a free Rx.com coupon.
What are the common side effects of Cholestyramine? ▼
Common side effects of Cholestyramine may include: Constipation, Stomach pain, Bloating, Gas, Nausea. This is not a complete list — consult your pharmacist or doctor for full side effect information.
Is there a generic version of Cholestyramine? ▼
Generic versions may be available for Cholestyramine. Generics contain the same active ingredients as brand-name drugs and are typically 80–90% cheaper. Search Cholestyramine on Rx.com to compare generic and brand prices at pharmacies near you.
What is the cheapest pharmacy for Cholestyramine? ▼
The cheapest pharmacy for Cholestyramine depends on your location and dosage. Rx.com compares prices at CVS, Walgreens, Walmart, Kroger, Costco, and thousands of independent pharmacies. Enter your ZIP code on Rx.com to find the lowest price for Cholestyramine near you.

Cholestyramine Coupons & Prices

Cholestyramine 378GM of 4GM/DOSE

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Cholestyramine Can — prescription drug image
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Cholestyramine 378gm of 4gm/dose (1)
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